Le, Truong-Giang; Pham, Hoai-Thu; Martin, James P.; Chataigner, Isabelle; Renaud, Jean-Luc published an article in 2020, the title of the article was Organocatalyzed regioselective and enantioselective synthesis of 1,4- and 1,2-dihydropyridines.Electric Literature of 79815-20-6 And the article contains the following content:
Herein, the first examples of asym. organocatalyzed synthesis of 1,2-dihydropyridines, affording enantioselective access to and partially solving regioselectivity challenges in the synthesis of dihydropyridines is reported. It has been demonstrated that through modification of organocatalysts both 1,2- and 1,4-dihydropyridines (1,2- and 1,4-DHPs) can be obtained with high regioselectivity (ratio of 1,2-DHP/1,4-DHP from 95/5 to 0/100) and enantioselectivity (33% ee for 1,2-DHPs and up to 98% ee for 1,4-DHPs) in good yields (up to 87%). The experimental process involved the reaction of H-Idc-OH(cas: 79815-20-6).Electric Literature of 79815-20-6
The Article related to dihydropyridine preparation green chem regioselective enantioselective organocatalyst, Heterocyclic Compounds (One Hetero Atom): Pyridines and other aspects.Electric Literature of 79815-20-6
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Indole alkaloid derivatives as building blocks of natural products from Bacillus thuringiensis and Bacillus velezensis and their antibacterial and antifungal activity study,
Preparation of Indole Containing Building Blocks for the Regiospecific Construction of Indole Appended Pyrazoles and Pyrroles